Diboron-Catalyzed Dehydrative Amidation of Aromatic Carboxylic Acids with Amines

DOI HANDLE Web Site Web Site 14 Citations 68 References Open Access

Abstract

Tetrakis(dimethylamido)diboron and tetrahydroxydiboron are herein reported as new catalysts for the synthesis of aryl amides by catalytic condensation of aromatic carboxylic acids with amines. The developed protocol is both simple and highly efficient over a broad range of substrates. This method thus represents an attractive approach for the use of diboron catalysts in the synthesis of amides without having to resort to stoichiometric or additional dehydrating agents.

Journal

  • Organic Letters

    Organic Letters 20 (15), 4397-4400, 2018-08-03

    ACS Publications

Citations (14)*help

See more

References(68)*help

See more

Related Projects

See more

Keywords

Details

Report a problem

Back to top