Formal [4 + 1]-Cycloaddition of Homopropargyl Alcohols to Diazo Dicarbonyl Compounds Giving Substituted Tetrahydrofurans

  • Fumiya Urabe
    Graduate School of Biomedical Sciences, Nagasaki University, Nagasaki 852-8521, Japan
  • Shohei Miyamoto
    Graduate School of Biomedical Sciences, Nagasaki University, Nagasaki 852-8521, Japan
  • Keisuke Takahashi
    Graduate School of Biomedical Sciences, Nagasaki University, Nagasaki 852-8521, Japan
  • Jun Ishihara
    Graduate School of Biomedical Sciences, Nagasaki University, Nagasaki 852-8521, Japan
  • Susumi Hatakeyama
    Graduate School of Biomedical Sciences, Nagasaki University, Nagasaki 852-8521, Japan

書誌事項

公開日
2014-01-13
資源種別
journal article
DOI
  • 10.1021/ol403746r
  • 10.1002/chin.201429120
公開者
American Chemical Society (ACS)

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説明

<jats:title>Abstract</jats:title><jats:p>This novel ring closure reaction involves tandem OH insertion/Conia‐ene cyclization under cooperative Rh(II)/Zn(II) catalysis, providing access to substituted tetrahydrofurans with complete (E)‐selection in the case of nonterminal alkynes (XII).</jats:p>

収録刊行物

  • Organic Letters

    Organic Letters 16 (3), 1004-1007, 2014-01-13

    American Chemical Society (ACS)

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