Antibody-Mediated Delivery of Chimeric BRD4 Degraders. Part 1: Exploration of Antibody Linker, Payload Loading, and Payload Molecular Properties

  • Peter S. Dragovich
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Thomas H. Pillow
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Robert A. Blake
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Jack D. Sadowsky
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Emel Adaligil
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Pragya Adhikari
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Sunil Bhakta
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Nicole Blaquiere
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Jinhua Chen
    WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
  • Josefa dela Cruz-Chuh
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Karen E. Gascoigne
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Steven J. Hartman
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Mingtao He
    Pharmaron Beijing, Co. Ltd., 6 Tai He Road, BDA, Beijing 100176, China
  • Susan Kaufman
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Tracy Kleinheinz
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Katherine R. Kozak
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Liang Liu
    Pharmaron Beijing, Co. Ltd., 6 Tai He Road, BDA, Beijing 100176, China
  • Liling Liu
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Qi Liu
    Pharmaron Beijing, Co. Ltd., 6 Tai He Road, BDA, Beijing 100176, China
  • Ying Lu
    WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
  • Fanwei Meng
    Pharmaron Beijing, Co. Ltd., 6 Tai He Road, BDA, Beijing 100176, China
  • Melinda M. Mulvihill
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Aimee O’Donohue
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Rebecca K. Rowntree
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Leanna R. Staben
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Steven T. Staben
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • John Wai
    WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
  • Jian Wang
    WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
  • BinQing Wei
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Catherine Wilson
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Jianfeng Xin
    Pharmaron Beijing, Co. Ltd., 6 Tai He Road, BDA, Beijing 100176, China
  • Zijin Xu
    WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
  • Hui Yao
    WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
  • Donglu Zhang
    Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
  • Hongyan Zhang
    WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
  • Hao Zhou
    WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
  • Xiaoyu Zhu
    WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China

収録刊行物

被引用文献 (2)*注記

もっと見る

詳細情報 詳細情報について

問題の指摘

ページトップへ