Antibody-Mediated Delivery of Chimeric BRD4 Degraders. Part 1: Exploration of Antibody Linker, Payload Loading, and Payload Molecular Properties
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- Peter S. Dragovich
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Thomas H. Pillow
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Robert A. Blake
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Jack D. Sadowsky
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Emel Adaligil
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Pragya Adhikari
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Sunil Bhakta
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Nicole Blaquiere
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Jinhua Chen
- WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
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- Josefa dela Cruz-Chuh
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Karen E. Gascoigne
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Steven J. Hartman
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Mingtao He
- Pharmaron Beijing, Co. Ltd., 6 Tai He Road, BDA, Beijing 100176, China
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- Susan Kaufman
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Tracy Kleinheinz
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Katherine R. Kozak
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Liang Liu
- Pharmaron Beijing, Co. Ltd., 6 Tai He Road, BDA, Beijing 100176, China
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- Liling Liu
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Qi Liu
- Pharmaron Beijing, Co. Ltd., 6 Tai He Road, BDA, Beijing 100176, China
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- Ying Lu
- WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
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- Fanwei Meng
- Pharmaron Beijing, Co. Ltd., 6 Tai He Road, BDA, Beijing 100176, China
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- Melinda M. Mulvihill
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Aimee O’Donohue
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Rebecca K. Rowntree
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Leanna R. Staben
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Steven T. Staben
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- John Wai
- WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
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- Jian Wang
- WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
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- BinQing Wei
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Catherine Wilson
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Jianfeng Xin
- Pharmaron Beijing, Co. Ltd., 6 Tai He Road, BDA, Beijing 100176, China
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- Zijin Xu
- WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
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- Hui Yao
- WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
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- Donglu Zhang
- Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States
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- Hongyan Zhang
- WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
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- Hao Zhou
- WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
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- Xiaoyu Zhu
- WuXi AppTec, 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, China
収録刊行物
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- Journal of Medicinal Chemistry
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Journal of Medicinal Chemistry 64 (5), 2534-2575, 2021-02-17
American Chemical Society (ACS)