Discovery of GBT440, an Orally Bioavailable R-State Stabilizer of Sickle Cell Hemoglobin

  • Brian Metcalf
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Chihyuan Chuang
    Cytokinetics, Inc., South San Francisco, California 94080, United States
  • Kobina Dufu
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Mira P. Patel
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Abel Silva-Garcia
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Carl Johnson
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Qing Lu
    Cytokinetics, Inc., South San Francisco, California 94080, United States
  • James R. Partridge
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Larysa Patskovska
    Albert Einstein College of Medicine, Bronx, New York 10461, United States
  • Yury Patskovsky
    Albert Einstein College of Medicine, Bronx, New York 10461, United States
  • Steven C. Almo
    Albert Einstein College of Medicine, Bronx, New York 10461, United States
  • Matthew P. Jacobson
    Department of Pharmaceutical Chemistry, University of California, San Francisco, California 94158, United States
  • Lan Hua
    Department of Pharmaceutical Chemistry, University of California, San Francisco, California 94158, United States
  • Qing Xu
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Stephen L. Gwaltney
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Calvin Yee
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Jason Harris
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Bradley P. Morgan
    Cytokinetics, Inc., South San Francisco, California 94080, United States
  • Joyce James
    Cytokinetics, Inc., South San Francisco, California 94080, United States
  • Donghong Xu
    Cytokinetics, Inc., South San Francisco, California 94080, United States
  • Athiwat Hutchaleelaha
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Kumar Paulvannan
    Tandem Sciences, Inc., Menlo Park, California 94025, United States
  • Donna Oksenberg
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
  • Zhe Li
    Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States

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