Discovery of GBT440, an Orally Bioavailable R-State Stabilizer of Sickle Cell Hemoglobin
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- Brian Metcalf
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Chihyuan Chuang
- Cytokinetics, Inc., South San Francisco, California 94080, United States
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- Kobina Dufu
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Mira P. Patel
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Abel Silva-Garcia
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Carl Johnson
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Qing Lu
- Cytokinetics, Inc., South San Francisco, California 94080, United States
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- James R. Partridge
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Larysa Patskovska
- Albert Einstein College of Medicine, Bronx, New York 10461, United States
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- Yury Patskovsky
- Albert Einstein College of Medicine, Bronx, New York 10461, United States
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- Steven C. Almo
- Albert Einstein College of Medicine, Bronx, New York 10461, United States
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- Matthew P. Jacobson
- Department of Pharmaceutical Chemistry, University of California, San Francisco, California 94158, United States
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- Lan Hua
- Department of Pharmaceutical Chemistry, University of California, San Francisco, California 94158, United States
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- Qing Xu
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Stephen L. Gwaltney
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Calvin Yee
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Jason Harris
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Bradley P. Morgan
- Cytokinetics, Inc., South San Francisco, California 94080, United States
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- Joyce James
- Cytokinetics, Inc., South San Francisco, California 94080, United States
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- Donghong Xu
- Cytokinetics, Inc., South San Francisco, California 94080, United States
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- Athiwat Hutchaleelaha
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Kumar Paulvannan
- Tandem Sciences, Inc., Menlo Park, California 94025, United States
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- Donna Oksenberg
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
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- Zhe Li
- Global Blood Therapeutics, Inc., South San Francisco, California 94080, United States
収録刊行物
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- ACS Medicinal Chemistry Letters
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ACS Medicinal Chemistry Letters 8 (3), 321-326, 2017-02-11
American Chemical Society (ACS)