In Silico and In Cell Hybrid Selection of Nonrapalog Ligands to Allosterically Inhibit the Kinase Activity of mTORC1
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- Raef Shams
- Emergent Bioengineering Materials Research Team, RIKEN Center for Emergent Matter Science, RIKEN, Wako, Saitama 351-0198, Japan
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- Akihiro Matsukawa
- Graduate School of Medicine, Dentistry, and Pharmaceutical Sciences, Okayama University, 2-5-1, Shikata, Kita-ku, 700-8558 Okayama, Japan
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- Yukari Ochi
- Graduate School of Medicine, Dentistry, and Pharmaceutical Sciences, Okayama University, 2-5-1, Shikata, Kita-ku, 700-8558 Okayama, Japan
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- Yoshihiro Ito
- Emergent Bioengineering Materials Research Team, RIKEN Center for Emergent Matter Science, RIKEN, Wako, Saitama 351-0198, Japan
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- Hideyuki Miyatake
- Department of Life Science, Graduate School of Science and Engineering, Saitama University, Saitama City, Saitama 338-8570, Japan
Journal
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- Journal of Medicinal Chemistry
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Journal of Medicinal Chemistry 65 (2), 1329-1341, 2021-06-30
American Chemical Society (ACS)
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Keywords
Details 詳細情報について
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- CRID
- 1360576118800171648
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- ISSN
- 15204804
- 00222623
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- Data Source
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- Crossref
- KAKEN