Light-induced control of protein destruction by opto-PROTAC

  • Jing Liu
    Department of Pathology, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA 02215, USA.
  • He Chen
    Mount Sinai Center for Therapeutics Discovery, Departments of Pharmacological Sciences and Oncological Sciences, Tisch Cancer Institute, Icahn School of Medicine at Mount Sinai, New York, NY 10029, USA.
  • Leina Ma
    Department of Pathology, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA 02215, USA.
  • Zhixiang He
    Department of Cancer Biology, Dana-Farber Cancer Institute, Boston, MA 02215, USA.
  • Dong Wang
    Department of Pathology, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA 02215, USA.
  • Yi Liu
    Department of Pathology, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA 02215, USA.
  • Qian Lin
    Department of Pathology, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA 02215, USA.
  • Tinghu Zhang
    Department of Cancer Biology, Dana-Farber Cancer Institute, Boston, MA 02215, USA.
  • Nathanael Gray
    Department of Cancer Biology, Dana-Farber Cancer Institute, Boston, MA 02215, USA.
  • H. Ümit Kaniskan
    Mount Sinai Center for Therapeutics Discovery, Departments of Pharmacological Sciences and Oncological Sciences, Tisch Cancer Institute, Icahn School of Medicine at Mount Sinai, New York, NY 10029, USA.
  • Jian Jin
    Mount Sinai Center for Therapeutics Discovery, Departments of Pharmacological Sciences and Oncological Sciences, Tisch Cancer Institute, Icahn School of Medicine at Mount Sinai, New York, NY 10029, USA.
  • Wenyi Wei
    Department of Pathology, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA 02215, USA.

説明

<jats:p> Opto-PROTAC adds a light-inducible switch on PROTAC, enabling optical control for targeted degradation of proteins of interest <jats:monospace>.</jats:monospace> </jats:p>

収録刊行物

  • Science Advances

    Science Advances 6 (8), eaay5154-, 2020-02-21

    American Association for the Advancement of Science (AAAS)

被引用文献 (5)*注記

もっと見る

詳細情報 詳細情報について

問題の指摘

ページトップへ