Discovery of Novel Azetidine Amides as Potent Small-Molecule STAT3 Inhibitors

  • Christine Brotherton-Pleiss
    Cancer Biology Program, University of Hawaii Cancer Center, University of Hawaii, Manoa, Honolulu, Hawaii 96813, United States
  • Peibin Yue
    Cancer Biology Program, University of Hawaii Cancer Center, University of Hawaii, Manoa, Honolulu, Hawaii 96813, United States
  • Kayo Nakamura
    Department of Chemistry, University of Hawaii, Manoa, 2545 McCarthy Mall, Honolulu, Hawaii 9682, United States
  • Weiliang Chen
    Department of Chemistry, University of Hawaii, Manoa, 2545 McCarthy Mall, Honolulu, Hawaii 9682, United States
  • Wenzhen Fu
    Cancer Biology Program, University of Hawaii Cancer Center, University of Hawaii, Manoa, Honolulu, Hawaii 96813, United States
  • Casie Kubota
    Cancer Biology Program, University of Hawaii Cancer Center, University of Hawaii, Manoa, Honolulu, Hawaii 96813, United States
  • Jasmine Chen
    Cancer Biology Program, University of Hawaii Cancer Center, University of Hawaii, Manoa, Honolulu, Hawaii 96813, United States
  • Felix Alonso-Valenteen
    Department of Biomedical Sciences, Cedars-Sinai Medical Center, Los Angeles, California 90048, United States
  • Simoun Mikhael
    Department of Biomedical Sciences, Cedars-Sinai Medical Center, Los Angeles, California 90048, United States
  • Lali Medina-Kauwe
    Department of Biomedical Sciences, Cedars-Sinai Medical Center, Los Angeles, California 90048, United States
  • Marcus A. Tius
    Cancer Biology Program, University of Hawaii Cancer Center, University of Hawaii, Manoa, Honolulu, Hawaii 96813, United States
  • Francisco Lopez-Tapia
    Cancer Biology Program, University of Hawaii Cancer Center, University of Hawaii, Manoa, Honolulu, Hawaii 96813, United States
  • James Turkson
    Cancer Biology Program, University of Hawaii Cancer Center, University of Hawaii, Manoa, Honolulu, Hawaii 96813, United States

書誌事項

公開日
2020-12-22
権利情報
  • https://pubs.acs.org/page/policy/authorchoice_ccbyncnd_termsofuse.html
DOI
  • 10.1021/acs.jmedchem.0c01705
公開者
American Chemical Society (ACS)

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