Structural Basis of Covalent Inhibitory Mechanism of TMPRSS2-Related Serine Proteases by Camostat

  • Gaohui Sun
    College of Chemistry, Fuzhou University, Fuzhou, Fujian, People’s Republic of China
  • Yaqun Sui
    College of Chemistry, Fuzhou University, Fuzhou, Fujian, People’s Republic of China
  • Yang Zhou
    College of Chemistry, Fuzhou University, Fuzhou, Fujian, People’s Republic of China
  • Junlin Ya
    College of Chemistry, Fuzhou University, Fuzhou, Fujian, People’s Republic of China
  • Cai Yuan
    College of Biological Science and Engineering, Fuzhou University, Fuzhou, Fujian, People’s Republic of China
  • Longguang Jiang
    College of Chemistry, Fuzhou University, Fuzhou, Fujian, People’s Republic of China
  • Mingdong Huang
    College of Chemistry, Fuzhou University, Fuzhou, Fujian, People’s Republic of China

書誌事項

公開日
2021-09-09
権利情報
  • https://doi.org/10.1128/ASMCopyrightv2
  • https://journals.asm.org/non-commercial-tdm-license
DOI
  • 10.1128/jvi.00861-21
公開者
American Society for Microbiology

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説明

<jats:p>Serine proteases are a large family of enzymes critical for multiple physiological processes and proven diagnostic and therapeutic targets in several clinical indications. The serine protease transmembrane protease serine 2 (TMPRSS2) was recently found to mediate SARS-CoV-2 entry into the host.</jats:p>

収録刊行物

  • Journal of Virology

    Journal of Virology 95 (19), e00861-21-, 2021-09-09

    American Society for Microbiology

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