Recent Advances in Transition‐metal‐catalyzed C−C Bond Formation via C(<i>sp</i><sup><i>2</i></sup>)−F Bond Cleavage

  • Liyan Fu
    Graduate School of Natural Science and Technology Okayama University 3-1-1 Tsushimanaka Kita-ku Okayama 700-8530 Japan
  • Qiang Chen
    Graduate School of Natural Science and Technology Okayama University 3-1-1 Tsushimanaka Kita-ku Okayama 700-8530 Japan
  • Yasushi Nishihara
    Research Institute for Interdisciplinary Science Okayama University 3-1-1 Tsushimanaka Kita-ku Okayama 700-8530 Japan

書誌事項

公開日
2021-04-14
権利情報
  • http://onlinelibrary.wiley.com/termsAndConditions#vor
DOI
  • 10.1002/tcr.202100053
公開者
Wiley

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説明

<jats:title>Abstract</jats:title><jats:p>The activation of a carbon‐fluorine bond is one of the most challenging topics in modern synthetic organic chemistry due to their low reactivity compared to other carbon‐halogen bonds. In this review, we present the recent developments since 2015 on cross‐coupling reactions that form C−C bonds via cleavage of C(<jats:italic>sp</jats:italic><jats:sup><jats:italic>2</jats:italic></jats:sup>)−F bonds. Not only the conventional activation of C(<jats:italic>sp</jats:italic><jats:sup><jats:italic>2</jats:italic></jats:sup>)−F bonds, but also decarbonylative or carbonyl‐retentive cleavage of C(acyl)−F bonds will be introduced. This paper mainly describes new protocols for the formation of C(<jats:italic>sp</jats:italic><jats:sup>2</jats:sup>)−C(<jats:italic>sp</jats:italic><jats:sup>3</jats:sup>), C(<jats:italic>sp</jats:italic><jats:sup>2</jats:sup>)−C(<jats:italic>sp</jats:italic><jats:sup>2</jats:sup>), and C(<jats:italic>sp</jats:italic><jats:sup>2</jats:sup>)−C(<jats:italic>sp</jats:italic>) bonds via transition‐metal‐catalyzed cleavage of C(<jats:italic>sp</jats:italic><jats:sup>2</jats:sup>)−F bonds.</jats:p>

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