The Nrf2/HO‐1 Axis in Cancer Cell Growth and Chemoresistance

書誌事項

公開日
2015-11-30
権利情報
  • http://creativecommons.org/licenses/by/4.0/
DOI
  • 10.1155/2016/1958174
公開者
Wiley

この論文をさがす

説明

<jats:p>The transcription factor, nuclear factor erythroid 2 p45‐related factor 2 (Nrf2), acts as a sensor of oxidative or electrophilic stresses and plays a pivotal role in redox homeostasis. Oxidative or electrophilic agents cause a conformational change in the Nrf2 inhibitory protein Keap1 inducing the nuclear translocation of the transcription factor which, through its binding to the antioxidant/electrophilic response element (ARE/EpRE), regulates the expression of antioxidant and detoxifying genes such as heme oxygenase 1 (HO‐1). Nrf2 and HO‐1 are frequently upregulated in different types of tumours and correlate with tumour progression, aggressiveness, resistance to therapy, and poor prognosis. This review focuses on the Nrf2/HO‐1 stress response mechanism as a promising target for anticancer treatment which is able to overcome resistance to therapies.</jats:p>

収録刊行物

被引用文献 (8)*注記

もっと見る

問題の指摘

ページトップへ