Highly Enantioselective Synthesis of Cyclopropylamine Derivatives via Ru(II)-Pheox-Catalyzed Direct Asymmetric Cyclopropanation of Vinylcarbamates

  • Soda Chanthamath
    Department of Environmental and Life Sciences, Toyohashi University of Technology, 1-1 Hibarigaoka, Tempaku-cho, Toyohashi 441-8580, Japan
  • Dao Thi Nguyen
    Department of Environmental and Life Sciences, Toyohashi University of Technology, 1-1 Hibarigaoka, Tempaku-cho, Toyohashi 441-8580, Japan
  • Kazutaka Shibatomi
    Department of Environmental and Life Sciences, Toyohashi University of Technology, 1-1 Hibarigaoka, Tempaku-cho, Toyohashi 441-8580, Japan
  • Seiji Iwasa
    Department of Environmental and Life Sciences, Toyohashi University of Technology, 1-1 Hibarigaoka, Tempaku-cho, Toyohashi 441-8580, Japan

書誌事項

公開日
2013-01-29
DOI
  • 10.1021/ol303404c
  • 10.1002/chin.201327047
公開者
American Chemical Society (ACS)

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説明

<jats:title>Abstract</jats:title><jats:p>This is the first report of the successful enantioselective carbene transfer cyclopropanation of diazoester into vinylcarbamate.</jats:p>

収録刊行物

  • Organic Letters

    Organic Letters 15 (4), 772-775, 2013-01-29

    American Chemical Society (ACS)

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