Boc<sub>3</sub>Arg-Linked Ligands Induce Degradation by Localizing Target Proteins to the 20S Proteasome
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- Yuntao Shi
- Graduate Program in Chemistry, ‡Graduate Program in Biochemistry and Biophysics, §Department of Biology, ∥Graduate Program in Molecular and Cell Biology, Brandeis University, Waltham, Massachusetts, United States
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- Marcus J.C. Long
- Graduate Program in Chemistry, ‡Graduate Program in Biochemistry and Biophysics, §Department of Biology, ∥Graduate Program in Molecular and Cell Biology, Brandeis University, Waltham, Massachusetts, United States
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- Masha M. Rosenberg
- Graduate Program in Chemistry, ‡Graduate Program in Biochemistry and Biophysics, §Department of Biology, ∥Graduate Program in Molecular and Cell Biology, Brandeis University, Waltham, Massachusetts, United States
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- Shican Li
- Graduate Program in Chemistry, ‡Graduate Program in Biochemistry and Biophysics, §Department of Biology, ∥Graduate Program in Molecular and Cell Biology, Brandeis University, Waltham, Massachusetts, United States
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- Aimee Kobjack
- Graduate Program in Chemistry, ‡Graduate Program in Biochemistry and Biophysics, §Department of Biology, ∥Graduate Program in Molecular and Cell Biology, Brandeis University, Waltham, Massachusetts, United States
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- Philip Lessans
- Graduate Program in Chemistry, ‡Graduate Program in Biochemistry and Biophysics, §Department of Biology, ∥Graduate Program in Molecular and Cell Biology, Brandeis University, Waltham, Massachusetts, United States
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- Rory T. Coffey
- Graduate Program in Chemistry, ‡Graduate Program in Biochemistry and Biophysics, §Department of Biology, ∥Graduate Program in Molecular and Cell Biology, Brandeis University, Waltham, Massachusetts, United States
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- Lizbeth Hedstrom
- Graduate Program in Chemistry, ‡Graduate Program in Biochemistry and Biophysics, §Department of Biology, ∥Graduate Program in Molecular and Cell Biology, Brandeis University, Waltham, Massachusetts, United States
収録刊行物
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- ACS Chemical Biology
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ACS Chemical Biology 11 (12), 3328-3337, 2016-10-18
American Chemical Society (ACS)