First Example of Phosphoramidate Approach Applied to a 4‘-Substituted Purine Nucleoside (4‘-Azidoadenosine): Conversion of an Inactive Nucleoside to a Submicromolar Compound versus Hepatitis C Virus
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- Plinio Perrone
- Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK, and Roche Palo Alto, 3431 Hillview Avenue, Palo Alto, California 94304
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- Felice Daverio
- Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK, and Roche Palo Alto, 3431 Hillview Avenue, Palo Alto, California 94304
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- Rocco Valente
- Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK, and Roche Palo Alto, 3431 Hillview Avenue, Palo Alto, California 94304
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- Sonal Rajyaguru
- Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK, and Roche Palo Alto, 3431 Hillview Avenue, Palo Alto, California 94304
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- Joseph A. Martin
- Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK, and Roche Palo Alto, 3431 Hillview Avenue, Palo Alto, California 94304
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- Vincent Lévêque
- Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK, and Roche Palo Alto, 3431 Hillview Avenue, Palo Alto, California 94304
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- Sophie Le Pogam
- Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK, and Roche Palo Alto, 3431 Hillview Avenue, Palo Alto, California 94304
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- Isabel Najera
- Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK, and Roche Palo Alto, 3431 Hillview Avenue, Palo Alto, California 94304
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- Klaus Klumpp
- Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK, and Roche Palo Alto, 3431 Hillview Avenue, Palo Alto, California 94304
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- David B. Smith
- Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK, and Roche Palo Alto, 3431 Hillview Avenue, Palo Alto, California 94304
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- Christopher McGuigan
- Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3XF, UK, and Roche Palo Alto, 3431 Hillview Avenue, Palo Alto, California 94304
収録刊行物
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- Journal of Medicinal Chemistry
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Journal of Medicinal Chemistry 50 (22), 5463-5470, 2007-10-03
American Chemical Society (ACS)