Covalent Ligand Screening Uncovers a RNF4 E3 Ligase Recruiter for Targeted Protein Degradation Applications

  • Carl C. Ward
    Department of Molecular and Cell Biology, University of California, Berkeley, Berkeley, California 94720, United States
  • Jordan I. Kleinman
    Novartis-Berkeley Center for Proteomics and Chemistry Technologies, University of California, Berkeley, Berkeley, California 94720, United States
  • Scott M. Brittain
    Novartis-Berkeley Center for Proteomics and Chemistry Technologies, University of California, Berkeley, Berkeley, California 94720, United States
  • Patrick S. Lee
    Novartis-Berkeley Center for Proteomics and Chemistry Technologies, University of California, Berkeley, Berkeley, California 94720, United States
  • Clive Yik Sham Chung
    Novartis-Berkeley Center for Proteomics and Chemistry Technologies, University of California, Berkeley, Berkeley, California 94720, United States
  • Kenneth Kim
    Department of Molecular and Cell Biology, University of California, Berkeley, Berkeley, California 94720, United States
  • Yana Petri
    Novartis-Berkeley Center for Proteomics and Chemistry Technologies, University of California, Berkeley, Berkeley, California 94720, United States
  • Jason R. Thomas
    Novartis-Berkeley Center for Proteomics and Chemistry Technologies, University of California, Berkeley, Berkeley, California 94720, United States
  • John A. Tallarico
    Novartis-Berkeley Center for Proteomics and Chemistry Technologies, University of California, Berkeley, Berkeley, California 94720, United States
  • Jeffrey M. McKenna
    Novartis-Berkeley Center for Proteomics and Chemistry Technologies, University of California, Berkeley, Berkeley, California 94720, United States
  • Markus Schirle
    Novartis-Berkeley Center for Proteomics and Chemistry Technologies, University of California, Berkeley, Berkeley, California 94720, United States
  • Daniel K. Nomura
    Department of Molecular and Cell Biology, University of California, Berkeley, Berkeley, California 94720, United States

書誌事項

公開日
2019-05-06
権利情報
  • https://doi.org/10.15223/policy-029
  • https://doi.org/10.15223/policy-037
  • https://doi.org/10.15223/policy-045
DOI
  • 10.1021/acschembio.8b01083
公開者
American Chemical Society (ACS)

この論文をさがす

収録刊行物

  • ACS Chemical Biology

    ACS Chemical Biology 14 (11), 2430-2440, 2019-05-06

    American Chemical Society (ACS)

被引用文献 (8)*注記

もっと見る

詳細情報 詳細情報について

問題の指摘

ページトップへ