Protein Degradation via CRL4<sup>CRBN</sup> Ubiquitin Ligase: Discovery and Structure–Activity Relationships of Novel Glutarimide Analogs That Promote Degradation of Aiolos and/or GSPT1

  • Joshua D. Hansen
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Kevin Condroski
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Matthew Correa
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • George Muller
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Hon-Wah Man
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Alexander Ruchelman
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Weihong Zhang
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Fan Vocanson
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Tim Crea
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Wei Liu
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Gang Lu
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Frans Baculi
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Laurie LeBrun
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Afshin Mahmoudi
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Gilles Carmel
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Matt Hickman
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States
  • Chin-Chun Lu
    Celgene Corporation, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States

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