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- Bernardini Raffaella
- Cell Therapeutics Inc.
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- Oliva Ambrogio
- Cell Therapeutics Inc.
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- Paganelli Alessandro
- Cell Therapeutics Inc.
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- Menta Ernesto
- EOS S.p.A. (Ethical Oncology Science)
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- Grugni Mario
- Cell Therapeutics Inc.
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- Munari Sergio De
- Cell Therapeutics Inc.
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- Goldoni Luca
- Cell Therapeutics Inc.
書誌事項
- 公開日
- 2009
- DOI
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- 10.1246/cl.2009.750
- 公開者
- 公益社団法人 日本化学会
この論文をさがす
説明
Boronic esters are key intermediates in the synthesis of biologically active compounds such as thrombin and proteasome inhibitors. However, they have low hydrolytic stability both during synthetic reactions and in biological media. We report the preparation of several boronic esters and a comparative study of their stability to hydrolysis vs. the corresponding pinanediol boronic esters, which are among the most hydrolytically stable. We discovered that the boronic esters derived from (1,1′-bicyclohexyl)-1,1′-diol are the most stable among those examined.
収録刊行物
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- Chemistry Letters
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Chemistry Letters 38 (7), 750-751, 2009
公益社団法人 日本化学会
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詳細情報 詳細情報について
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- CRID
- 1390282679562055808
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- NII論文ID
- 10025124576
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- NII書誌ID
- AA00603318
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- ISSN
- 13480715
- 03667022
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- 本文言語コード
- en
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- データソース種別
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- JaLC
- Crossref
- CiNii Articles
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- 抄録ライセンスフラグ
- 使用不可