Synthesis and Antifungal Activity of 5-Methoxy-2-nitrophenylphosphoramidothioates
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- KOHSAKA Hideo
- Pesticides Research Laboratory, Takarazuka Research Center, Sumitomo Chemical Co., Ltd.
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- OGURI Yukio
- Pesticides Research Laboratory, Takarazuka Research Center, Sumitomo Chemical Co., Ltd.
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- SASAKI Mitsuru
- Pesticides Research Laboratory, Takarazuka Research Center, Sumitomo Chemical Co., Ltd.
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- MUKAI Kunio
- Pesticides Research Laboratory, Takarazuka Research Center, Sumitomo Chemical Co., Ltd.
Bibliographic Information
- Other Title
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- 5-メトキシ-2-ニトロフェニルチオノリン酸アミド類の合成と抗菌活性
- 5-メトキシー2-ニトロフェニルチオノリン酸アミド類の合成と抗菌活性〔英文〕
- 5 メトキシ 2 ニトロフェニルチオノリンサン アミドルイ ノ ゴウセイ ト
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Abstract
Thirty-three 5-methoxy-2-nitrophenylphosphoramidothioates and phosphonamidothioates were synthesized and tested for their antifungal activity against downy mildew on cucumber in greenhouse pot tests. Among the compounds O-ethyl O-(5-methoxy-2-nitrophenyl) phosphoramidothioates having either an isopropylamino group, a 1-cyano-2-propylamino group, a 1-methoxy-2-butylamino group, or a s-butylamino group showed the highest activity. A 1-methoxy-2-propylamino group, a 3-methoxypropylamino group and a 1, 1-dioxotetrahydrothiophen-3-ylamino group effectively reduced the phytotoxicity without affecting the antifungal activity. Among N-isopropylphosphoramidothioates and phosphonamidothioates, O-methyl or O-ethyl phosphoramidothioates showed the highest activity. Chloromethylphosphonamidothioate was also effective, but phenylphosphonamidothioate was not effective. O-Ethyl O-(5-methoxy-2-nitrophenyl) N-s-butylphosphoramidate was hardly effective.
Journal
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- Journal of Pesticide Science
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Journal of Pesticide Science 12 (3), 415-419, 1987
Pesticide Science Society of Japan
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Details 詳細情報について
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- CRID
- 1390282680187888896
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- NII Article ID
- 110001712100
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- NII Book ID
- AN00196227
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- ISSN
- 03851559
- 13490923
- 1348589X
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- NDL BIB ID
- 3146546
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- Data Source
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- JaLC
- IRDB
- NDL
- Crossref
- NDL-Digital
- CiNii Articles
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- Abstract License Flag
- Disallowed