Cyclization, Ring‐Expansion, and Several Cascade Reactions Utilizing Allenylic Molecular Structure Characteristics

書誌事項

タイトル別名
  • Cyclization, Ring-Expansion, and Several Cascade Reactions Utilizing Allenylic Molecular Structure Characteristics

この論文をさがす

説明

Various kinds of new reactions based on allenylic molecular structure characteristics have been described. Specifically, mild alkaline hydrolysis of diethyl α-acetylamino (or methoxy) -α-alkynylmalonates generates conjugated allenyl esters which promote 5-endo-mode heterocyclic cyclization giving trisubsutituted oxazoles, SH-enzyme inhibition, new chiral pyrrolinones (cathepsin B inhibitors) formation, and Myers-type biradical aromatization in a cascade reaction manner. Systematic ortho vicinal-endo-mode-, geminal spiro-endo-mode-, and meta ansa-endo-mode-cyclization reactions have been accomplished by using numerous conjugated allenyl ketones and Lewis acids. Base-mediated and palladium (0) -catalyzed cascade heterocyclic and carbocyclic ring-expansion reactions have been achieved by using hydroxy-substituted allenyl cyclic compounds.

収録刊行物

被引用文献 (1)*注記

もっと見る

参考文献 (48)*注記

もっと見る

キーワード

詳細情報 詳細情報について

問題の指摘

ページトップへ