Dual Catalysis with Copper and Rhenium for Trifluoromethylation of Propargylic Alcohols: Efficient Synthesis of α‐Trifluoromethylated Enones

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Published
2014-07-30
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  • http://onlinelibrary.wiley.com/termsAndConditions#vor
DOI
  • 10.1002/chem.201403447
  • 10.1002/chin.201511092
Publisher
Wiley

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<jats:title>Abstract</jats:title><jats:p>Trifluoromethylation of propargylic alcohols to provide (<jats:italic>Z</jats:italic>)‐α‐trifluoromethylated enones and β‐unsubstituted α‐trifluoromethylated enones proceeded with high yield and selectivity in the presence of CuI/Re<jats:sub>2</jats:sub>O<jats:sub>7</jats:sub>. The <jats:italic>Z</jats:italic> isomer was formed under kinetic control, though it is less stable than the <jats:italic>E</jats:italic> isomer in terms of steric repulsion.</jats:p>

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