EI-1941-1 and -2, Novel Interleukin-1.BETA. Converting Enzyme Inhibitors Produced by Farrowia sp. E-1941: I. Biochemical Characterization of EI-1941-1 and -2

  • KOIZUMI FUMITO
    Tokyo Research Laboratories, Kyowa Hakko Kogyo Co., Ltd.
  • MATSUDA YUZURU
    Tokyo Research Laboratories, Kyowa Hakko Kogyo Co., Ltd. Corporate Planning Department, Kyowa Hakko Kogyo Co., Ltd.
  • NAKANISHI SATOSHI
    Tokyo Research Laboratories, Kyowa Hakko Kogyo Co., Ltd. Strategic Planning Department, Pharmaceuticals Company, Kyowa Hakko Kogyo Co., Ltd.

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タイトル別名
  • I. Biochemical Characterization of EI-1941-1 and-2

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説明

EI-1941-1 and -2 isolated from the culture broths of Farrowia sp. selectively inhibited the human recombinant ICE activity with IC50 values of 0.086 and 0.006μM, respectively, without inhibiting elastase and cathepsin B. EI-1941-1 and -2 also inhibited mature interleukin-1β secretion from THP-1 cells induced by LPS with IC50 values of 5.0 and 10.3μM, respectively. Biochemical characterizations of EI-1941-1 and-2 are described in this article.

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詳細情報 詳細情報について

  • CRID
    1390282679125269504
  • NII論文ID
    130003504074
  • DOI
    10.7164/antibiotics.56.464
  • COI
    1:CAS:528:DC%2BD3sXktlyjtbs%3D
  • ISSN
    18811469
    00218820
  • PubMed
    12870812
  • 本文言語コード
    en
  • 資料種別
    journal article
  • データソース種別
    • JaLC
    • Crossref
    • PubMed
    • CiNii Articles
  • 抄録ライセンスフラグ
    使用不可

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